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Talabostat mesylate

CAS No. 150080-09-4

Talabostat mesylate ( Val-boroPro (mesylate); PT100 (mesylate )

Catalog No. M17326 CAS No. 150080-09-4

Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Talabostat mesylate
  • Note
    Research use only, not for human use.
  • Brief Description
    Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.
  • Description
    Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein. This agent may also stimulate the production of colony stimulating factors, such as granulocyte colony-stimulating factor (G-CSF), resulting in the stimulation of hematopoiesis.
  • Synonyms
    Val-boroPro (mesylate); PT100 (mesylate
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phosphatase
  • Recptor
    DPP-4
  • Research Area
    Metabolic Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    150080-09-4
  • Formula Weight
    310.18
  • Molecular Formula
    C10H23BN2O6S
  • Purity
    98%
  • Solubility
    DMSO : ≥ 40 mg/mL. 128.96 mM
  • SMILES
    OB([C@H]1N(C(=O)[C@@H](N)C(C)C)CCC1)O.CS(=O)(=O)O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Cristillo AD, et al. HIV-1 Env vaccine comprised of electroporated DNA and protein co-administered with Talabostat. Biochem Biophys Res Commun. 2008 May 23;370(1):22-6.
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