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Talabostat mesylate
CAS No. 150080-09-4
Talabostat mesylate ( Val-boroPro (mesylate); PT100 (mesylate )
Catalog No. M17326 CAS No. 150080-09-4
Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 88 | In Stock |
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| 10MG | 143 | In Stock |
|
| 50MG | 357 | In Stock |
|
| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameTalabostat mesylate
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NoteResearch use only, not for human use.
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Brief DescriptionTalabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.
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DescriptionTalabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein. This agent may also stimulate the production of colony stimulating factors, such as granulocyte colony-stimulating factor (G-CSF), resulting in the stimulation of hematopoiesis.
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SynonymsVal-boroPro (mesylate); PT100 (mesylate
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PathwayMetabolic Enzyme/Protease
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TargetPhosphatase
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RecptorDPP-4
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Research AreaMetabolic Disease
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Indication——
Chemical Information
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CAS Number150080-09-4
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Formula Weight310.18
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Molecular FormulaC10H23BN2O6S
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Purity98%
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SolubilityDMSO : ≥ 40 mg/mL. 128.96 mM
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SMILESOB([C@H]1N(C(=O)[C@@H](N)C(C)C)CCC1)O.CS(=O)(=O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Cristillo AD, et al. HIV-1 Env vaccine comprised of electroporated DNA and protein co-administered with Talabostat. Biochem Biophys Res Commun. 2008 May 23;370(1):22-6.
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